ICI-199,441
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| Systematic (IUPAC) name | |
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2-(3,4-dichlorophenyl)-N-methyl-N-[(1S)-1-phenyl-2-pyrrolidin-1-ylethyl]acetamide
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| Identifiers | |
| CAS Number | 115199-84-3  |
| PubChem | CID: 3082718 |
| ChEMBL | CHEMBL38576  |
| Chemical data | |
| Formula | C21H24Cl2N2O |
| Molecular mass | 391.333 g/mol |
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ICI-199,441 is a drug which acts as a potent and selective κ-opioid agonist, and has analgesic effects.[1][2] It is a biased agonist of the KOR, and is one of a relatively few KOR ligands that is G protein-biased rather than β-arrestin-biased.[1]
See also
References
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