C-8813

C-8813

Systematic (IUPAC) name
trans-4-(p-Bromophenyl)-4-(dimethylamino)-1-(2-(thiophen-2-yl)ethyl)cyclohexanol
Identifiers
CAS Number	616898-54-5 N
PubChem	CID: 11058633
Chemical data
Formula	C20H26BrNOS
Molecular mass	408.394 g/mol
SMILES BrC1=CC=C([C@@]2(CC[C@](CC2)(CCC3=CC=CS3)O)N(C)C)C=C1
NY (what is this?)  (verify)

C-8813 (thiobromadol) is a potent μ-opioid receptor agonist with a distinctive chemical structure which is not closely related to other established families of opioid drugs. The trans-isomer was found to be around 591 times more potent than morphine in animal studies. The same study assigned a potency of 504 times that of morphine to the related compound BDPC.

C-8813 is claimed to be similarly potent at the δ-opioid receptor, which antagonizes the mu depression of breathing, presumably making the drug safer.

C-8813 has never been used in humans.

See also

• BDPC
• Ciramadol
• Faxeladol
• Profadol
• Tapentadol
• Tramadol